Conjugate hydrotrifluoromethylation of α,β-unsaturated acyl-oxazolidinones: synthesis of chiral fluorinated amino acids.

نویسندگان

  • Holger Erdbrink
  • Ilona Peuser
  • Ulla I M Gerling
  • Dieter Lentz
  • Beate Koksch
  • Constantin Czekelius
چکیده

A novel conjugate hydrofluoroalkylation of α,β-unsaturated acyl-oxazolidinones is described. Using this method, enantiomerically pure β-trifluoromethylated amino acids were prepared. Trifluorovaline and trifluoroisoleucine were incorporated into peptides and found to show extremely low α-helix propensities.

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عنوان ژورنال:
  • Organic & biomolecular chemistry

دوره 10 43  شماره 

صفحات  -

تاریخ انتشار 2012